Biochem/physiol Actions
Primary Targetk opioid receptor
General description
A highly potent and selective non-alkaloid positive allosteric modulator of κ-opioid receptors (Ki = 4.3 nM and 16 nM for native and cloned κ-opioid receptors, respectively). Also acts as a D2DR partial agonist (Ki = 5-10 nM). Used in studies of addition.
Legal Information
CALBIOCHEM is a registered trademark of Merck KGaA, Darmstadt, Germany
Packaging
1 mg in Glass bottle
Warning
Toxicity: Standard Handling (A)
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